{"id":870,"date":"2026-01-23T23:01:26","date_gmt":"2026-01-23T21:01:26","guid":{"rendered":"https:\/\/www.transtoyou.com\/lt\/product\/candesartan\/"},"modified":"2026-02-13T13:51:46","modified_gmt":"2026-02-13T11:51:46","slug":"candesartanas","status":"publish","type":"product","link":"https:\/\/www.transtoyou.com\/lt\/product\/candesartanas\/","title":{"rendered":"Kandesartanas"},"content":{"rendered":"<p>Kandesartanas yra angiotenzino II receptori\u0173 blokatorius (ARB), kuris taikosi \u012f vien\u0105 i\u0161 pagrindini\u0173 organizmo kraujosp\u016bd\u017eio hormon\u0173. Angiotenzinas II paprastai prisijungia prie AT1 receptori\u0173 lygiuosiuose raumenyse, dengian\u010diuose arterijas, nurodydamas jiems susitraukti ir skatindamas antinks\u010dius i\u0161skirti aldosteron\u0105, kuris savo ruo\u017etu ver\u010dia inkstus kaupti drusk\u0105 ir vanden\u012f. S\u0117d\u0117damas tuose pa\u010diuose receptoriuose, kandesartanas blokuoja \u0161\u012f signal\u0105: kraujagysl\u0117s i\u0161lieka atsipalaidavusios, skys\u010di\u0173 susilaikymas ma\u017e\u0117ja, o kraujosp\u016bdis suma\u017e\u0117ja be kosulio, kuris gali varginti ACE inhibitorius.<\/p>\n<p>Nurytas, prodrug kandesartanas cileksetilis greitai vir\u0161kinimo trakte konvertuojamas \u012f aktyv\u0173 kandesartan\u0105. Maksimalios koncentracijos pasiekiamos per 34 valandas, o molekul\u0117s tvirtas prisijungimas prie receptori\u0173 suteikia jai galutin\u012f pusin\u0117s eliminacijos period\u0105 9 valandos, ta\u010diau antihipertenzinis poveikis trunka vis\u0105 dien\u0105, tod\u0117l vienkartinis dozavimas yra patogus.<\/p>\n<p>Dideliuose LIFE ir CHARM tyrimuose kandesartanas suma\u017eino insulto, \u0161irdies sm\u016bgio ir \u0161irdies nepakankamumo hospitalizacijas, palyginti su beta blokatoriais ar placebu. Sistoliniame \u0161irdies nepakankamume jis da\u017enai derinamas su beta blokatoriais ir mineralokortikoid\u0173 antagonistais, kad suma\u017eint\u0173 skilveli\u0173 sieneli\u0173 stres\u0105 ir pagerint\u0173 i\u0161gyvenamum\u0105.<\/p>\n<p>Kandesartanas gerai toleruojamas: galvos svaigimas arba nedideli inkst\u0173 funkcijos poky\u010diai yra pagrindiniai ankstyvieji nepageidaujami rei\u0161kiniai, o serumo kalio lygis paprastai pakyla tik \u0161iek tiek. Kadangi jis yra labai selektyvus, jis netrukdo bradikininui; tod\u0117l angioedema yra reta, o plau\u010diai i\u0161lieka \u0161var\u016bs.<\/p>\n<p>Tablet\u0117s yra pl\u0117vele dengtus, \u012fpjautus ir stabilios iki 30 \u00b0C, tod\u0117l jas patogu ve\u017etis. \u017dmon\u0117ms, ie\u0161kantiems \u0161velnaus, nuolatinio kraujosp\u016bd\u017eio kontrol\u0117s arba ACE inhibitoriaus alternatyvos, kandesartanas suteikia \u012frodyt\u0105 \u0161irdies ir kraujagysli\u0173 apsaug\u0105 su minimaliu gyvenimo b\u016bdo sutrikdymu.<\/p>\n","protected":false},"excerpt":{"rendered":"<ul>\n<li>24 valand\u0173 kraujosp\u016bd\u017eio apsauga<\/li>\n<li>Be kosulio, ACE laisvas komfortas<\/li>\n<li>Klinikiniu b\u016bdu \u012frodytas insulto suma\u017einimas<\/li>\n<\/ul>\n","protected":false},"featured_media":872,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[136],"product_tag":[],"expert":[21],"class_list":{"0":"post-870","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-aukstas-kraujo-spaudimas","7":"expert-dr-m-sharoyko","9":"first","10":"instock","11":"shipping-taxable","12":"product-type-variable"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.0 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Candesartanas | Kraujo Spaudimo Lengv\u0117jimas - Transtoyou<\/title>\n<meta name=\"description\" content=\"Candesartanas: Blokuok kraujosp\u016bd\u017eio hormonus su \u0161iuo ARB. 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